Description

[Cys2, Tyr3,Orn5,Pen7]. This somatostatin analog is a very potent and highly selective ligand for m-opioid receptors.

SEQUENCE: H-DPhe-Cys-Tyr-DTrp-Orn-Thr-Pen-Thr-NH2 (trifluoroacetate salt)
(Cys2 and Pen7 Bridge)

ONE-LETTER SEQUENCE: DPhe-CY-DTrp-Orn-T-Pen-T-NH2 (Cys2 and Pen7 Bridge)

MOLECULAR FORMULA: C₅₀H₆₈N₁₁O₁₁S₂

MOLECULAR WEIGHT: 1063.3

STORAGE CONDITIONS: -20 ± 5 °C

CAS REGISTRY NUMBER: [103429-31-8]

SYNONYMS:

RESEARCH AREA: Pain

REFERENCES:
K.N.Hawkins et al., J. Pharmacol. Exp. Ther., 248, 73 (1989)
K.Gulya et al., Eur. J. Pharmacol., 150, 355 (1988)
L.F. Tseng et al., The Journal of Pharmacol. and Experim. Therap., 280, 600 (1997)

SKU(s): SOMA-005A, SOMA-005B

KEYWORDS: hormone